| Sl. No. | Name | Title of Ph.D. Thesis | University | Year |
| 1. | A. V. Narender Reddy
(Co-guidance) | Synthesis of Nitrogen Heterocycles of Potential Biological Interest: Fused 1,2,4-Benzothiadiazine-1,1-Dioxide | Osmania | 1986 |
| 2. | B. S. P. Reddy | Synthesis and Biological Evaluation of a New Class of 5-Thio pyrrolo[2,1-c] [1,4]benzodiazepine Antitumour Antibiotics | Osmania | 1995 |
| 3. | N. Venugopal Rao | Synthesis and Biological Study for DNA Interactive New Type of pyrrolo[2,1-c][1,4] Benzodiazepine Antitumour Antibiotics | Osmania | 1996 |
| 4. | Y. Damayanthi | Biotransformations in the Synthesis of Some Biologically Active Compounds | Osmania | 1997 |
| 5. | M. Venkateswara Rao | Enzymes as Biocatalysts in the Synthesis of Biologically Active Compounds | Osmania | 1997 |
| 6. | Ms. N. L. Gayatri | Synthesis of Podophyllotoxin Lignans as DNA Topoisomerase Inhibitors | Osmania | 1999 |
| 7. | Mr. B. S. N. Reddy | Design and Synthesis of New Anthramycin Class of Compounds as DNA Binding Antitumour Antibiotics | Osmania | 1999 |
| 8. | E. Laxman | Design and Synthesis of Novel podophyllotoxin Dimers and DNA interactive Pyrrolo [2,1-c][1,4] Benzodiazepine Antitumour Antibiotics | Osmania | 2000 |
| 9. | N. Laxman | Design, Synthesis and Biological Activity of New Class of C8-Linked Pyrrolo[2,1-c][1,4] Benzodiazepines | Osmania | 2001 |
| 10. | Md. Arifuddin | Development of Methodologies for the opening of oxiranes: Regenation of Carbonyl Compounds and Synthesis of New Podophyllotoxin Congeners as Anticancer Agents | Osmania | 2001 |
| 11. | G. Suresh Kumar Reddy | Design and Combinatorial Synthesis of Pyrrolobenzodiazepine Antitumour Antibiotics | Osmania | 2002 |
| 12. | K. Venkata Ramana | Chemoenzymatic Synthesis of some Biologically Active Compounds | Osmania | 2003 |
| 13. | G. Ramesh | Design and Synthesis of DNA Interactive Novel Pyrrolo[2,1-c][1,4] benzodiazepine Antitumour Antibiotics and Preparation of 4-b-arylamino Podophyllotoxin Congeners | Kakatiya | 2003 |
14. | G. B. Ramesh Khanna | Chemoenzymatic Synthesis of Optically pure β-hydroxy nitriles and their Application towards the Preparation of Biologically Important Comounds | Osmania | 2004 |
| 15. | P. Ramulu | Design and Synthesis of Novel Pyrrolo[2,1-c][1,4]benzodiazepine dimers and its C8-linked Hybrids as DNA Interactive Compounds | Kakatiya | 2004 |
| 16. | P.S.M.M. Reddy | Design and Synthesis of DNA Cross-linking new Pyrrolo[2,1-c] [1,4]benzodiazepine Dimers as Antitumor Antibiotics | Andhra | 2004 |
| 17. | Mahendra Sandbhor | Chemoenzymatic Synthesis of Biologically Important Compounds by One-pot Lipase Resolution Protocol | Pune | 2004 |
| 18. | O. Srinivas | Synthesis and Biological Evaluation of C2 and C8 linked Novel Dimers and Hybrids of pyrrolo[2,1-c][1,4] benzodiazepine as DNA-binding Antitumour Antibiotics | Osmania | 2005 |
| 19. | R. Ramu | Design and Synthesis of New Pyrrolo[2,1-c][1,4]benzodiazepine Hybrids as DNA Interactive Antitumour Agents | Kakatiya | 2005 |
| 20. | Gagan Chouhan | Catalytic and Biocatalytic Transformations in Ionic Liquid: Synthesis of Some Biologically Important Compounds | Pune | 2006 |
| 21. | K. Laxma Reddy | Combinatorial Synthesis of Pyrrolobenzodiazepine Antibiotics | Osmania | 2006 |
| 22. | A. V. Ramana | Design, Synthesis and Anticancer Evaluation of Novel Pyrrolo[2,1-c][1,4]benzodiazepine Hybrids, Chrysin Conjugates and Preparation of some Bioactive Heterocycles | Nagarjuna | 2006 |
| 23. | A. Hari Babu | Design, Synthesis and Biological Evaluation of Pyrrolo[2,1-c][1,4]benzodiazepine hybrids and phenazine analogues | Kakatiya | 2006 |
| 24. | Ahmad Ali Shaik | Chemoenzymatic Synthesis of Biologically Active entities and Development of Thiolactomycin Based Compounds as New Antitubercular Agents | Osmania | 2006 |
| 25. | D. Rajasekhar Reddy | Design and Synthesis of DNA-binding Pyrrolo[2,1-c][1,4]benzodiazepine Conjugates and Development of New Synthetic Methodologies | S. V. Univ. | 2006 |
| 26. | B. Ashwini Kumar | Synthesis and Biological Activity of New Podophyllotoxin Congeners and C8-linked DNA Interactive Pyrrolo[2,1-c][1,4]benzodiazepines | Osmania | 2006 |
| 27. | K. Srinivas Reddy | Design, Synthesis and Biological Evaluation of Novel Benzodiazepine Analogues and Pyrrolo[2,1-c][1,4] benzodiazepine Hybrids | Osmania | 2006 |
| 28. | V.Devaiah | Synthesis and Biological activity of Novel pyrrolobenzodiazepine Hybrids and Combinatorial Synthesis of Biologically active Nitrogen Heterocycles | Kakatiya | 2006 |
| 29. | B. Rajendra Prasad | Design and Synthesis of Novel Pyrrolo[2,1-c] [1,4]benzodiazepine Hybrids and related Compounds as Potential Anticancer Agents | Kakatiya | 2007 |
| 30. | Kaleem Ahmed | Synthesis and Biological Evaluation of Benzodiathiadiazens and Antibubercular Drugs | Osmania | 2007 |
| 31. | T. Venkatesh | Design, Synthesis and Activity Studies of New Pyrrolo[2,1-c][1,4]Benzodiazepine Prodrugs and Hybrids | S. V. Univ. | 2007 |
| 32. | Mr. T. Krishnaji | Chemoenzymatic Synthesis of biologically important compounds | Nagarjuna | 2007 |
| 33. | Mr. N. Shankaraiah | Synthesis of DNA-Interactive C2/C8-linked Pyrrolo [2,1-c][1,4]benzodiazepine Hybrids and Combinatorial Synthesis of itsDimers / Hybrids and Bioactive fused [2,1-b] Quinazolinones | Kakatiya | 2007 |
| 34. | Mr. Md. Naseer Ahmed Khan | New Pyrrolo[2,1-c][1,4] Benzodiazepine: Synthesis and Biological Evaluation | Kakatiya | 2007 |
| 35. | Mr. P. Praveen Kumar | Design, Synthesis and Biological Evolution of Novel substituted Benzimidazole derivatives linked to C8 position of Pyrrolo [2,1-c][1,4]Benzodiazepine Conjugates | Nagarjuna | 2008 |
| 36. | Mr. M. S. Malik | Synthesis of biologically active compounds and application of biocatalysts in the preparation of chiral entities | Osmania | 2009 |
| 37. | Mr. K. Srikanth | Design and synthesis of DNA cross-linking novel C-8 linked pyrrolo[2,1-c][1,4]benzodiazepine antitumour antibiotics | Nagarjuna | 2009 |
| 38. | Mr. G. Balakishan | Design, synthesis and biological activity of a new class of C-8 linked pyrrolo[2,1-c][1,4] benzodiazepine analogues as antitumour antibiotics | Nagarjuna | 2009 |
| 39. | Mr. Mohd. Ameeruddin | Synthesis of Biologically Active Chiral Compounds Employing Catalytic & Enzymatic Processes | Kakatiya | 2012 |
| 40. | Mr. Shaik Azeeza | Design and Synthesis of New Molecules based on Thiolactomycin as Potential Antitubercular, Antimalarial Agents and Enantioselective Synthesis of (3R,4R), (3S,4S)-dihydroxypyrrolidines | Nagarjuna | 2010 |
| 41. | Mr. Rajesh V.C.R.M.C. Shetty | Design, Synthesis and Bioactive Studies of Caboline, Cabazole and Fluorenes linked to Pyrrolo[2,1-c] [1,4] benzodiazepines and Deve -lopment of New Methodologies | Kakatiya | 2010 |
| 42. | Ms. E. Vijaya Bharathi | Synthesis and Biological Evaluation of New Hybrids of Pyrrolo[2,1-c][1,4] benzodiazepines and Quinazolinones as Potential Anticancer agents | Osmania | 2010 |
| 43. | Mr. Syed Farooq Adil | Synthesis of Pharmacologically important compounds using biotransformation | JNTU | 2007 |
| 44. | Mr. Rajendar | Design, Synthesis and Biological Activity of DNA-interactive Novel Pyrrolo[2,1-c][1,4] benzodiazepines | Osmania | 2012 |
| 45. | Ms. Rohini | Epoxide hydrolase and its application in Biotransformations | Nagarjuna | ------ |
| 46. | Mr. J.Surendranadha Reddy | Synthesis and biolgocial activity of isoxazole linked pyrrolo[2,1-c] [1,4]benzodiazepines as DNA interactive compounds | S. V. Univ. | 2010 |
| 47. | Mr. Dastagiri | Design, synthesis and bioactive studies of pyrrolo[2,1-c][1,4] benzodiazepine linked to pyrazole and imadazole | S. V. Univ. | 2010 |
| 48. | Mr. P. Suresh | Design and synthesis of podophyllotoxin anticancer agents as congeners | Kakatiya | 2012 |
| 49. | Mr. S. Prabhakar | Design, synthesis and biological evaluation of new pyrrolo[2,1-c][1,4]benzodiazepines and their dimers by employing ‘click’ chemistry | Kakatiya | 2012 |
| 50. | Mr. A. Malla Reddy | Synthesis and biological evaluation of pyrrolobenzodiazepines as antitumour antibiotics | Kakatiya | 2012 |
| 51. | M. Kashi Reddy | Design and synthesis of naphthalene and pyridine linked pyrrolobenzodiazepine hybrids as anticancer antibiotics | Kakatiya | 2012 |
| 52. | Mr. Y. V. V. Srikanth | Synthesis of bisindole conjugates and 2-anilinonicotinyl linked oxadiazoles/2-aminobenzothiazoles/triazolobenzo-thiadiazines | Nagarjuna | 2012 |
| 53. | Mr. P. Venkat Reddy | Development of new approaches for some bioactive lactone natural products and spiroacetals–aculeatins | Osmania | 2011 |
| 54. | Mr. A. Viswanath | Synthesis and biological evaluation of new pyrrolobenzodiazepines. Tetrazoles and quinazolinone derivatives as potential anticancer agents | Nagarjuna | 2012 |
| 55. | Mr. J. N. S. R. Murthy | Synthesis and biological evaluation of new class of pyrolo[2,1-c][1,4]napthodiazepines and flavones | Nagarjuna | 2013 |
| 56. | Mr. P. Raju | Synthesis of prodrugs based on pyrrolobenzodiazepines as selective anticancer agents | JNTU | ------- |
| 57. | Mr. Ratna Reddy | Synthesis and Biological Evaluation of Combretastatin A-4 and Benzophenone Hybrids as Antimitotic Agents | S. V. Univ. | 2015 |
| 58. | Mr. Nagaseshadri | Synthesis and anti cancer potential of indolin-2-one conjugates of beta-carboline, benzimidazole and indole and n-sulfonyl indolyl glyoxylamides | S. V. Univ. | 2016 |
| 59. | Mr. G. Ramakrishna | Design and synthesis of combretotostatin linked pyrrolo[2,1-c][1,4]benzodiaphine hybrids as antitumor antibiotics | S. V. Univ. | 2011 |
| 60. | Mr Jaki Rasheed Tamboli | Design and synthesis of podophyllotoxin analogues and their biological evaluation | JNTU | 2013 |
| 61. | Mr Shaikh Faazil Shaikh Raheem | Synthesis of nitrogen heterocyclic conjugates: potential chemotherapeutics for cancer and tuberculosis | Osmania | 2013 |
| 62. | Mrs P. Swapna | Synthesis of oxazolidinones and triazoles as antimicrobial compounds and imidazothiadiazoles as potential anticancer agents | JNTU | 2013 |
| 63. | Mr V. Santosh Reddy | Synthesis and anticancer activity of heterocycles based on the chalcone and 2-anilinopyridine/pyrazole/isoxazole congeners as a tubulin inhibitors | Osmania | 2013 |
| 64. | Mr N. V. Subba Reddy | Synthesis and anticancer potential of Benzofurans, 2 anilinopyridines and imidazopyridines and arylation of benzothiazoles | S.V. Univ. | 2014 |
| 65. | Mr. Bajee Shaik | Synthesis of new molecules based on combretastatin A-4, cinnamamide and 1,4-dihydropyridine scaffolds as potential anticancer agents | JNTU | 2016 |
| 66. | Mr. M. Balakrishna | Synthesis and anticancer potential of chalcones, cinnamides and picolinamide containing heterocycles: total synthesis of Synargentolide-A and Cytospolide-D | KU | 2014 |
| 67. | Ms. Farheen Sultana | Synthesis and anticancer activity of new pyrrolobenzodiazepine, quinazolinone, imidazobenzothiazole and chalcone derivatives | Osmania | 2013 |
| 68. | Mr. Md. Ashraf | Synthesis of 2-Anilinopyridine and Combretastatin Conjugates as Anticancer Agents | Osmania | 2014 |
| 69. | Mr. V. Sreenivasulu | Design, Synthesis and Anticancer Potential of Pyrroloquinolodiazepines, β-carboline Hybrids and Development of Greener Methodologies | JNTU | 2014 |
| 70. | Mr. G Bharath Kumar | Synthesis and biological evaluation of aminostilbene, phenstatin, isocombretastatin, imidazopyrimidine and isoxazoles conjugates as tubulin polymerization inhibitors | KU | 2015 |
| 71. | Mr. Mohd. Ali | New chemical entities based on nitrogen containing privileged heterocycles aspotential chemotherapeutic agents | Osmania | 2013 |
| 72. | Mr. Saidi Reddy | Total synthesis of nhatrangin a, lentiginosine, b-conhydrine, and podophyllotoxin congeners as anticancer agents | S.V. Univ. | 2014 |
| 73. A | Mr. A Venka Subba Rao | Synthesis and Biological evaluation of Heterocyclic Conjugates as Microtubule targeting Potential Anticancer Agent | AcSIR | 2015 |
| 74. | Mr. Anver Basha Shaik | Synthesis of pyrazole based conjugates as tubulin polymerization inhibitors | JNTU | 2015 |
| 75. | Mr. Praveen Kumar Reddy Adiyala | Synthesis of pyrrolo[2,1-c][1,4]benzodiazepine (PBD) prodrugs, development of new methods for synthesis of heterocyclic libraries and total synthesis of pinolide | Osmania | 2016 |
| 76. | Mr. P S Srikanth | Combretastatin/Quinoline Hybrids and Spiroquinazolines as Tubulin Polymerization Inhibitors | AcSIR | 2017 |
| 77. | Mr. Siddiq Pasha | Synthesis of Imidazo[2,1-b]thiazole and Benzo[d]imidazo[2,1-b]thiazole Conjugates as Potential Microtubule Targeting Agents | AcSIR | 2017 |
| 78. | Mr. Thoukhir Basha shaik | Biological implications of some new cytotoxic agents and development of microemulsion delivery systems | Nagarjuna | 2017 |
| 79. | Mr.Lakshma Nayak | Studies on the mechanism and Induction of Apoptosis by New Chemical Entities against Breast/Lung Cancer | JNTU | 2017 |
| 80. | Mr. N Shankar Rao | Cinnamide/Naphthalimide/Chalcone/Pyrazoline Hybrids as PotentialAnticancer Agents and Quinoline Derivatives as Antimicrobial Agents | AcSIR | 2017 |
| 81. | Mr.Rasala Mahesh | Synthesis and anticancer potential of trimethoxystyryl benzene sulfonamide/sulfonates, quinazolinone-urea, quinazolinone- arylpropenones and green synthesis of spirooxindole,phyrazolo-pyrimidine derivatives | Osmania | 2017 |
| 82. | Mr. M. Kishore | Design and development of indol and biphenyl linked heterocyclic as potent anticancer agents | Osmania | 2017 |
| 83. | Mr. Narasimha Reddy | Phenacyl azide: A versatile intermediate for the Synthesis of Imidazo[1,2-a]pyridines, Pyrrolo[1,2-a]imidazoles, β-Enaminoes, Pyrrolidin-2-ones and Amides; Diastereoselective Synthesis of Spiro[cyclopropane-1,3’-indolin]-2’-ones as potential Anticancer agents | Osmania | 2017 |
| 84. | Mr. M. Satish | Synthesis of b-carboline conjugates as DNA interactive topoisomerase inhibitiors and development of new synthetic methods | Osmania | 2017 |
| 85. | Mr. Bagul Chandrakanth Deoram | Synthesis and Biological Evaluation of Pyrazolo[1,5-α] pyrimidines and Triaryl Olefins as EGFR Inhibitors | NIPER-H | 2017 |
| 86. | Mr. Chander Singh Digwal | Application of Vanadyl Sulfate in the Development of newer Synthetic Methodologies and Preparation of 4-(Arylthiazol-2-yl)morpholines as Potential Cytotoxic Agents | NIPER-H | 2017 |
| 87. | Mr. M.P. Narasimha Rao | Synthesis and biological evaluation of β-carboline-benzimidazole and imidazothiadiazole and indole-indolinone conjugates as potential anticancer agents | Osmania | 2018 |
| 88. | Mr. N.Praveen Kumar | Design, Synthesis and Cytotoxicity Evaluation of Phenanthrene Hybrids and Novel Method for Functionalized Enamino-2-oxindoles | NIPER-H | 2018 |
| 89. | Mr. B.Nagaraju | Synthesis of Pyrazole, coumarinconjugates and their cytotoxicity: Development of greener methodologies for some biologically important heterocyclics. | AcSIR | 2018 |
| 90. | Mrs. K.Jeshma | Synthesis and biological evaluation of new β-carboline, coumarin and indole based conjugates and development of photocatalytic methodologies. | AcSIR | 2018 |
| 91. | Mr. T.Yellaiah | Synthesis of β-carboline and dihydrofuran congeners as potential anti cancer agents and development of new methodologies for biologically useful heterocyclics | AcSIR | 2018 |
| 92. | Mr. S.Satish | Synthesis of imidazopyridines, thienopyridines and aminopyridylacylamides as potential anticancer agents: Development of newer methodologies for the imidazopyridine scaffold. | AcSIR | 2018 |
| 93. | Mrs. Faria Sultana | Design synthesis and biological evaluation of hybrid hetrocyclic scaffolds as potential anticancer agents. | Osmania | 2018 |
| 94. | Mr.Ibrahim Bin Sayeed | Imidozothizole, imidazopyridine benoimdazothiazole linked propenonetriazole and oxindole as potent anti cancer agents. | AcSIR | 2018 |
| 95. | Mr.M.V.P.S. Vishnu Vardhan | Evaluation of antiproliferative activity and understanding the mode of action of some natural/synthetic molecules | JNTU | 2019 |
| 96. | Mr. K. Suresh Babu | Design and development of greener methods for the synthesis of heterocyclic compounds; Evaluation of their cytotoxicity and antimicrobial activity. | Osmania | 2019 |
| 97. f | Mr. Feroz | Synthesis of fused imidazoles and 2-methylquinoline conjugates as cytotoxici agents: Develpement of newer methods for fused imidazoles and benzimidazoles | AcSIR | 2019 |
| 98. | Mr. K. N. Visweswara Sastry | Development of new methodologies for the synthesis of Benzoxazocine triazoles, Pyrazole Conjugates, Trisubstituted Pyrazoles, Substituted Quinazolines, Polysubstituted Pyrroles and their Biological Evaluation | NIPER-H | 2019 |
| 99. | Mr. Namballa Hari Krishna | Design, Synthesis and Biological Evaluation of β-carboline-Cinnamate Conjugates as HDAC Inhibitors, Development of Domino Method for Carbazole Scaffolds, Total Synthesis of Mupirocin H and (-) Aspergillide C | NIPER-H | 2019 |
100. | Mrs. P. Venkata Sriramya | Synthesis of Curcumin Inspired Heterocyclic Analogues as Potent Cytotoxic Agents and Development of New Synthetic Methodologies | NIPER-H | 2019 |
| 101. | Mr. Abdul Rahim Abdul Rauf | Synthesis & Biological Evaluation of Indole, Isatin, Quinoline and Benzimidazole based Congeners as Anticancer and Antimicrobial Agents: Development of New Synthetic methodologies | AcSIR | 2019 |
| 102. | Ms. D. Kavitha | Design, synthesis and biological evaluation of biaryl fused oxindoles, cinnmamides, as antimotumor agents and novel method development for the synthesis of imidazoquinazolinones, benzimidazo-quinazolines an quinazolinones | NIPER-H | 2020 |
| 103. | Mrs. Jadala Chetna | Design, synthesis of CA4 linked β-carboline, chalcone, sulfonyl piperazine hybrids as antitumor agents and development of novel methodology for the synthesis of pyrroles | NIPER-H | 2020 |
| 104. | Ms.Yadav Upasana Rameshbhai | Synthesis and biological evaluation of heterocyclic hybrids | NIPER-H | 2020 |
| 105. | Mrs. Soma Gupta | Beta glucosidase from Bacillus stratosphericus SG9-Optimization, Production, Characterization and Application as efficient Biosurfactant producer | Nagarjuna | 2020 |
| 106. | Mrs. M. Geeta Sai Mani | Molecular iodine catalyzed synthesis of fused heterocycles via oxidative annulation and design, synthesis and biological evaluation of imidazo[1,5-a]pyriinyl 2-propenone derivatives as anticancer agents | NIPER-H | 2020 |
| 107. | Ms.R.Sunitha Rani | Studies on Extracellular Polymeric Substances from Marine Bacteria and their Applications | Nagarjuna | 2020 |
| 108. | Mr. Mohd. Adil Shareef | Synthesis and Bilogical studies of imidazo, indolo and indenopyrazole fused heterocyclics as potential chemotherapeutic agents | AcSIR | 2020 |
| 109. | Mr. B. Prasad | Design and synthesis of E7010 derivatives as anticancer agents and development of new organic methodologies | Osmania | 2020 |
| 110. | Mr. Prasanna Anjaneyulu Yakkala | Synthesis and development of heterocyclic hybrids as potential anticancer agents | Jamia Hamdard | |
| 111. | Mr. Anku Sharma | Synthesis of quinazolinone based anticancer agents targeting Wnt signalling | Jamia Hamdard | |